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"5AB-A<C6:8 4;O 287=0G5==O >4=>3> ?>:07=8:0 A5GV: :5B>=8. >=F5=B@0FVW @>1>G>3> @5035=BC: 5B>=8: =0B@VN =VB@>?@CAA84 4,9%. #<>28 715@V30==O: 2 IV;L=> 70:@8BV9 >@83V=0;L=V9 C?0:>2FV 2 ACE><C B5<=><C <VAFV 70 B5<?5@0BC@8 2V4 +2 4> +30 C.?0:45033696500-0-01>@0B>@=V @50:B82853462 "@83;VF5@848 "25001V@ @5035=BV2 ?@87=0G5=89 4;O :V;L:VA=>3> in vitro 287=0G5==O B@83;VF5@84V2 C A8@>20BFV V ?;07<V :@>2V ;N48=8. $0AC20==O: =5 <5=H5 R1:1x250 <;, R2 AB0=40@B: 1E3 <; !:;04 @5035=BV2: R1 CD5@ C4A0 (@ 7,2) 50 <<>;L/; 4-E;>@D5=>; 4 <<>;L/; Mg 2+ 15 <<>;L/; AT$ 2 <<>;L/; ;VF5@>;:V=070 e" 0,4 :4/; 5@>:A84070 e" 2 :4/; V?>?@>B5W=;V?070 e" 2 :4/; ;VF5@>;-3-D>AD0B>:A84070 e" 0,5 :4/; 4-0<V=>0=B8?V@8= 0,5 <<>;L/; R2 AB0=40@B :>=F5=B@0FVO 2:070=0 =0 D;0:>=V >5DVFVT=B ?5@5@0EC=:C (<3/4;) E 0,0113 = <<>;L/; >1>GV E0@0:B5@8AB8:8 =5 3V@H5 70: 'CB;82VABL: 9,74 <3/4; (0,11 <<>;L/;) V=V9=VABL: 4> 1062 <3/4; (12 <<>;L/;) V0?07>= 28<V@N20==O: 9,74  1062 <3/4; (0,11  12 <<>;L/;) #<>28 715@V30==O 2V4 +2 4> +8 C.?0:1033696500-0-01>@0B>@=V @50:B82853393%>;5AB5@8= % 100001V@ @5035=BV2 ?@87=0G5=89 4;O Vn vitro 287=0G5==O E>;5AB5@8=C C A8@>20BFV V ?;07<V :@>2V ;N48=8. $0AC20==O: =5 <5=H5 R1: 1 x 1000 <; @8=F8? <5B>4C 5B>4 @C=BCTBLAO =0 >A=>2V @>7@>1:8 ;;5=0 B0 V=., WW <>48DV:0FVW >H;0C, V7 ?>40;LH8<8 24>A:>=0;5==O<8 4;O ?V428I5==O AB01V;L=>ABV @5035=BC C @>7G8=0E !:;04 @5035=BV2: R1 CD5@ C4A0 50 <<>;L/; $5=>; 5 <<>;L/; 4-0<V=>0=B8?V@8= 0,3 <<>;L/; %>;5AB5@>;5AB5@070 e" 200 4/; %>;5AB5@>;>:A84070 e" 50 4/; 5@>:A84070 e" 3 k4/; >5DVFVT=B ?5@5@0EC=:C <3/4; E 0,026 = <<>;L/; >1>GV E0@0:B5@8AB8:8 =5 3V@H5 70: 'CB;82VABL 4,2 (<3/4;) (0,11 <<>;L/;) V=V9=VABL: 4> 695 (<3/4;) (18,07 <<>;L/;) V0?07>= 28<V@N20==O: 4,2 695 <3/4; (0,11 18,07 <<>;L/;) #<>28 715@V30==O 2V4 +2 4> +8 C.?0:633696500-0-01>@0B>@=V @50:B82859123$>AD>@ 25001V@ @5035=BV2 ?@87=0G5=89 4;O :V;L:VA=>3> in vitro 287=0G5==O D>AD>@C C A8@>20BFV V ?;07<V :@>2V, 0 B0:>6 C A5GV ;N48=8. $0AC20==O: =5 <5=H5 R1: 1 x 250 <;, R2 !B0=40@B: 1 x 5 <; @8=F8? <5B>4C 5>@30=VG=89 D>AD>@ C ?@8ACB=>ABV AV@G0=>W :8A;>B8 CB2>@NT V7 <>;V140B>< 0<<>=VN D>AD><>;V140B=89 :><?;5:A. >3;8=0==O :><?;5:AC =0 340 =< T ?@>?>@FV9=8< :>=F5=B@0FVW D>AD>@C C 7@07:>2V. !:;04 @5035=BV2 R1 <>=VN <>;V140B 1,0 <<>;L/; 8A;>B0 AV@G0=0 336 <<>;L/; R2 !B0=40@B :>=F5=B@0FVO 2:070=0 =0 D;0:>=V >5DVFVT=B ?5@5@0EC=:C <<>;L/; = 0,32 E <3/4; >1>GV E0@0:B5@8AB8:8 =5 3V@H5 70: 'CB;82VABL: 0,20 <3/4; (0,064 <<>;L/;) V=V9=VABL: 4> 22,9 <3/4; (7,40 <<>;L/;) V0?07>= 28<V@N20==O: 0,20 22,9 <3/4; (0,064 7,40 <<>;L/;). #<>28 715@V30==O 2V4 +2 4> +8 C.?0:233696500-0-01>@0B>@=V @50:B8285288303=V9 MG 25001V@ @5035=BV2 ?@87=0G5=89 4;O :V;L:VA=>3> in vitro 287=0G5==O <03=VN C A8@>20BFV V ?;07<V :@>2V, A?8==><>7:>2V9 @V48=V, 0 B0:>6 A5GV ;N48=8. $0AC20==O: =5 <5=H5 R1: 1 x 250 <;, R2 AB0=40@B: 1 E 5 <; 03=V9 C ;C6=><C A5@54>28IV CB2>@NT V7 :A8;V48;>28< A8=V< 7010@2;5=89 :><?;5:A, O:89 28<V@NNBL D>B><5B@8G=>. =B5=A82=VABL 7010@2;5==O T ?@>?>@FV9=>N :>=F5=B@0FVW <03=VN C 7@07:>2V. " 70AB>A>2CTBLAO O: @5035=B 4;O 7<5=H5==O 2?;82C :0;LFVN. !:;04 @5035=BV2 R1 A8;V48;>289 A8=V9 (I) 110 <:<>;L/; B0=>;0<V= 1 <>;L/; " 60 <:<>;L/; R2 AB0=40@B: :>=F5=B@0FVO 2:070=0 =0 D;0:>=V >5DVFVT=B ?5@5@0EC=:C <<>;L/; = 0,4114 E <3/4; >1>GV E0@0:B5@8AB8:8 =5 3V@H5 70: 'CB;82VABL: 0,16 <3/4; (0,064 <<>;L/;) V=V9=VABL: 4> 5,85 <3/4; (2,4 <<>;L/;) V0?07>= 28<V@N20==O: 0,16  5,85 <3/4; (0,064  2,4 <<>;L/;) #<>28 715@V30==O 2V4 +2 4> +8 C.?0:233696500-0-01>@0B>@=V @50:B828457890;LFV9 CA 25001V@ @5035=BV2 ?@87=0G5=89 4;O :V;L:VA=>3> in vitro 287=0G5==O :0;LFVN 2 A8@>20BFVV ?;07<V :@>2V, 0 B0:>6 C A5GV ;N48=8. $0AC20==O: =5 <5=H5 R1: 1 x 250 <;, R2 cB0=40@B: 1 x 5 <; @8=F8? <5B>4C @A5=07> III 7 V>=0<8 :0;LFVN ?@8 @H 6, 5 CB2>@NNBL :>;L>@>289 :><?;5:A, V=B5=A82=VABL 7010@2;5==O O:>3> T ?@>?>@FV9=>N :>=F5=B@0FVW V>=V2 :0;LFVN. 8<V@N20==O ?>3;8=0==O :><?;5:AC ?@>2>48BLAO =0 650 =< (650-660 =<). @A5=07> III <0T 25;8:C A?>@V4=5=VABL (k = 1 x 10-7) 4> V>=V2 :0;LFVN V =57=0G=C 4> V=H8E V>=V2, B><C V=HV :0BV>=8 A8@>20B:8, ?;07<8 V A5GV =5 2?;820NBL =0 @57C;LB0B8 287=0G5==O. !:;04 @5035=BV2: R1 @A5=07> III 0,10 <<>;L/; $>AD0B=89 1CD5@ (pH 7,8 0,1) 50 <<>;L/; R2 (AB0=40@B ) :>=F5=B@0FVO 2:070=0 =0 D;0:>=V >5DVFVT=B ?5@5@0EC=:C (<3/4;) E 0,25 = <<>;L/; >1>GV E0@0:B5@8AB8:8 =5 3V@H5 70: 'CB;82VABL: 0,6 <3/4; (0,15 <<>;L/;) V=V9=VABL: 4> 16 <3/4; (4,0 <<>;L/;) V0?07>= 28<V@N20==O: 0,6  16 <3/4; (0,15  4,0 <<>;L/;) #<>28 715@V30==O 2V4 +2 4> +8 C.?0:533696500-0-01>@0B>@=V @50:B82852924" - "/  " 50001V@ @5035=BV2 ?@87=0G5=89 4;O :V;L:VA=>3> in vitro 287=0G5==O "/" (ALT/GPT, 0;0=V=0<V=>B@0=AD5@078) C A8@>20BFV V ?;07<V :@>2V. $0AC20==O: =5 <5=H5 R1: 4 x 100 <;, R2: 1 E 100 <; "/" (ALT/GPT) V !"/" (AST/GOT)  =091V;LH 206;82V ?@54AB02=8:8 0<V=>B@0=AD5@07, I> :0B0;V7CNBL ?5@5B2>@5==O 0-:5B>:8A;>B =0 0<V=>:8A;>B8 H;OE>< ?5@5=>AC 0<V=>3@C?. !:;04 @5035=BV2: R1 "@VA-1CD5@ (pH 7,5) 137,5 <<>;L/; L-;0=V= 709 <<>;L/;  (<V:@>1=0) e" 2000 U/; R2 CAPSO 20 <<>;L/; 2-:A>3;CB0@0B 85 <<>;L/;  1,05 <<>;L/; >5DVFVT=B ?5@5@0EC=:C U/; E 0,017 = <::0B/; >1>GV E0@0:B5@8AB8:8 =5 3V@H5 70: 'CB;82VABL: 4,4 U/; (0,075 <::0B/;) V=V9=VABL: 4> 360 U/; (6,12 <::0B/;) V0?07>= 28<V@N20==O: 4,4 - 360 U/; (0,075 - 6,12 <::0B/;) #<>28 715@V30==O 2V4 +2 4> +8 C.?0:1033696500-0-01>@0B>@=V @50:B82852950!" - !"/" 50001V@ @5035=BV2 ?@87=0G5=89 4;O :V;L:VA=>3> in vitro 287=0G5==O 0A?0@B0B0<V=>B@0=AD5@078 (!") C A8@>20BFV V ?;07<V :@>2V ;N48=8. $0AC20==O: =5 <5=H5 R1: 4 x 100 <;, R2: 1 E 100 <; "/" (ALT/GPT) V !"/" (AST/GOT)  =091V;LH 206;82V ?@54AB02=8:8 0<V=>B@0=AD5@07, <VABOBLAO C 2AVE B:0=8=0E ;N48=8, ?>@V2=O=> 28A>:89 @V25=L A?>AB5@V30TBLAO 2 ?0@5=E8<V ?5GV=:8, =8@:>28E B:0=8=0E, C A5@F528E V A:5;5B=8E < O7>28E B:0=8=0E. !:;04 @5035=BV2: R1 "@VA-1CD5@ (pH 7,8) 110 <<>;L/; L-A?0@B0B 340 <<>;L/;  e" 4000 4/;  e" 750 4/; R2 CAPSO 20 <<>;L/; 2-:A>3;CB0@0B 85 <<>;L/;  1,05 <<>;L/; >5DVFVT=B ?5@5@0EC=:C 4/; E 0,017 = <::0B/; >1>GV E0@0:B5@8AB8:8 =5 3V@H5 70: 'CB;82VABL: 3,84 4/; (0,064 <::0B/;) V=V9=VABL: 390 4/; (5,1 <::0B/;) V0?07>= 28<V@N20==O: 3,84  390 4/; (0,064  5,1 <::0B/;) #<>28 715@V30==O 2V4 +2 4> +8 C.?0:1033696500-0-01>@0B>@=V @50:B82853030-;CB0<V;B@0=AD5@070 " 10001V@ @5035=BV2 ?@87=0G5=89 4;O in vitro 287=0G5==O 30<<0-3;CB0<V;B@0=AD5@078 (", GGT) C A8@>20BFV V ?;07<V :@>2V ;N48=8. $0AC20==O: =5 <5=H5 R1: 4 x 20 <;, R2: 1 E 20 <; @8=F8? <5B>4C V=5B8G=89 <5B>4 7 L--3;CB0<V;-3-:0@1>:AV-4-=VB@>0=V;V4>< (Persijn & van der Slik), AB0=40@B87>20=89 C 2V4?>2V4=>ABV 4> @5:><5=40FV9 IFCC. !:;04 @5035=BV2: R1 "@VA-1CD5@ (pH 8,25) 125 <<>;L/; ;VF8;3;VF8= 125 <<>;L/; R2 L--3;NB0<V;-3-:0@1>:AV-4-=VB@>0=V;V4 20 <<>;L/; >5DVFVT=B ?5@5@0EC=:C 4/; E 0,017 = <::0B/; >1>GV E0@0:B5@8AB8:8 =5 3V@H5 70: 'CB;82VABL: 1,68 4/; V=V9=VABL: 4> 500 4/; V0?07>= 28<V@N20==O: 1,68 - 500 4/; #<>28 715@V30==O 2V4 +2 4> +8 C?0:533696500-0-01>@0B>@=V @50:B828530720:B0B453V4@>35=070  10001V@ @5035=BV2 ?@87=0G5=89 4;O Vn vitro 287=0G5==O ;0:B0B453V4@>35=078, () C A8@>20BFV V ?;07<V :@>2V ;N48=8 (<5B>4 DGKCH). $0AC20==O: =5 <5=H5 R1: 4 x 20 <;, R2: 1 E 20 <; 5B>4 ?B8<V7>20=89 :V=5B8G=89 <5B>4 C 2V4?>2V4=>ABV 7 @5:><5=40FVO<8 DGKC (7 ?V@C20B><).  @5035=BV <VAB8BLAO ?V@C20B 73V4=> <5B>4C 5=@V B0 V=. !:;04 @5035=BV2: R1 "@VA-1CD5@ (pH 7,5) 100 <<>;L/; V@C20B 2,0 <<>;L/; R2  1,66 <<>;L/; >5DVFVT=B ?5@5@0EC=:C 4/; E 0,017 = <::0B/; >1>GV E0@0:B5@8AB8:8 =5 3V@H5 70: 'CB;82VABL: 43,8 4/; (0,746 <::0B/;) V=V9=VABL: 4> 1200 4/; (20,4 <::0B/;) V0?07>= 28<V@N20==O: 43,8 200 4/; (0,746 20,4 <::0B/;) #<>28 715@V30==O 2V4 +2 4> +8 C.?0:533696500-0-01>@0B>@=V @50:B82853590!5G>28=0 ' 25001V@ @5035=BV2 ?@87=0G5=89 4;O :V;L:VA=>3> in vitro 287=0G5==O A5G>28=8 C A8@>20BFV V ?;07<V :@>2V, 0 B0:>6 C A5GV ;N48=8 $0AC20==O: =5 <5=H5 R1: 4 x 50 <;, R2: 1 E 50 <;, R3 AB0=40@B: 1 E 5 <; @8=F8? <5B>4C V=5B8G=89 D5@<5=B0B82=89 <5B>4 ("0;:5-(C15@B0, 24>A:>=0;5=89 "VDD0=V) !:;04 @5035=BV2: R1 "@VA-1CD5@ 100 <<>;L/; -:5B>3;CB0@0B 5,49 <<>;L/; #@5070 (Jack Bean) > 10 :4/<;  (<V:@>1=0) > 3,8 :4/<; R2  1,66 <<>;L/; 50:FV9=>-=59B@0;L=V =0?>2=N20GV V AB01V;V70B>@8 R3 AB0=40@B :>=F5=B@0FVO 2:070=0 =0 D;0:>=V >5DVFVT=B ?5@5@0EC=:C <<>;L/; = 0,1665 E <3/4; !5G>28=0 (<3/4;) E 0,467 = 7>B A5G>28=8 (<3/4;) 7>B A5G>28=8 (<3/4;) E 2,14 = !5G>28=0 (<3/4;) >1>GV E0@0:B5@8AB8:8 =5 3V@H5 70: 'CB;82VABL: 11,5 <3/4; (1,91 <<>;L/;) V=V9=VABL: 4> 300 <3/4; (49,8 <<>;L/;) (A5G>28=0) 4> 140 <3/4; (23,24 <<>;L/;) (07>B A5G>28=8) V0?07>= 28<V@N20==O: 11,5 - 300 <3/4; (1,91  23,24 <<>;L/;) #<>28 715@V30==O 2V4 +2 4> +8 C.?0:1833696500-0-01>@0B>@=V @50:B82853586!5G>20 :8A;>B0   20001V@ @5035=BV2 ?@87=0G5=89 4;O :V;L:VA=>3> in vitro 287=0G5==O A5G>2>W :8A;>B8 2 A8@>20BFV V ?;07<V :@>2V, 0 B0:>6 C A5GV ;N48=8. $0AC20==O: =5 <5=H5 R1: 4 x 50 <;, R2 !B0=40@B: 1 x 5 <; !5G>20 :8A;>B0 T :V=F528< ?@>4C:B>< <5B01>;V7<C ?C@8=V2, =C:;5W=>28E :8A;>B V =C:;5>?@>B5W4V2. B65, 70=865==O 01> 7028I5==O @V2=O A5G>2>W :8A;>B8 A2V4G0BL ?@> ?>@CH5==O <5B01>;V7<C. !:;04 @5035=BV2: R1 Pipes-1CD5@ pH 7,0 50 <<>;L/; %$! 0,50 <<>;L/; #@8:070 e" 0,32 :4/; 5@>:A84070 e" 1,0 :4/; 4-0<V=>0=B8?V@8= 0,31 <<>;L/; * 3,5-4VE;>@-2-D5=>;AC;LD>=0B R2 !B0=40@B >=F5=B@0FVO 2:070=0 =0 D;0:>=V A5G>20 :8A;>Ba 357 <:<>;L/; >5DVFVT=B ?5@5@0EC=:C <3/4; E 60 = <:<>;L/; >1>GV E0@0:B5@8AB8:8 =5 3V@H5 70: 'CB;82VABL: 0,49 <3/4; (29,46 <:<>;L/;) V=V9=VABL: 4> 25 <3/4; (1475 <:<>;L/;) V0?07>= 28<V@N20==O: 0,49  25 <3/4; (29,46 - 1475 <:<>;L/;) #<>28 715@V30==O 2V4 +2 4> +8 C.?0:633696500-0-01>@0B>@=V @50:B82852928C6=0 D>AD0B070 $  150 5035=B ?@87=0G5=89 4;O in vitro 287=0G5==O ;C6=>W D>AD0B078 C A8@>20BFV V ?;07<V :@>2V ;N48=8. $0AC20==O: R1: 4 E 30 <;, R2: 1 x 30 <; @8=F8? @50:FVW # 2V4?>2V4=>ABV V7 @5:><5=40FVO<8 IFCC. 2-0<V=>-2-<5B8;-1-?@>?0=>; + ?0@0-=VB@>D5=V;D>AD0B + H2O !:;04 @5035=BV2: R1 2-0<V=>-2-<5B8;-1-?@>?0=>; () 1CD5@ @ 10,4 434 <<>;L/; 03=VN 0F5B0B 2,48 <<>;L/; &8=:C AC;LD0B 1,24 <<>;L/; HEDTA 2,48 <<>;L/; R2 p-?0@0=VB@>D5=V;D>AD0B 81,6 <<>;L/; >5DVFVT=B ?5@5@0EC=:C 4/; E 0,017 = <::0B/; >1>GV E0@0:B5@8AB8:8 =5 3V@H5 70: 'CB;82VABL: 4,5 4/; V=V9=VABL: 4> 1300 4/; V0?07>= 28<V@N20==O: 4,5 1300 4/; #<>28 715@V30==O 2V4 +2 4> +8 C?0:633696500-0-01>@0B>@=V @50:B82853395V?>?@>B5W= ) 80 01V@ @5035=BV2 ?@87=0G5=89 4;O in vitro 287=0G5==O ) E>;5AB5@8=C (HDL) C A8@>20BFV V ?;07<V :@>2V ;N48=8 $0AC20==O: =5 <5=H5 R1: 2 x 30 <;, R2: 2 E 10 <; @8=F8? <5B>4C PVS V PEGME, I> <VABOBLAO C A:;04V @5035=BC R1, CB2>@NNBL :><?;5:A V7 CAV<0 ;V?>?@>B5W40<8 (), ) V EV;><V:@>=0<8), >:@V< ). ><?;5:A 1;>:CT CG0ABL F8E ;V?>?@>B5W4V2 C D5@<5=B0B82=8E @50:FVOE ?@8 4>4020==V p5035=BC R2. %>;5AB5@8=5AB5@070 (%) V E>;5AB5@8=>:A84070 (%) C A:;04V R2 >:8A;NNBL BV;L:8 )-E>;5AB5@8=. 5@5:8A 2>4=N, I> CB2>@NTBLAO ?V4 G0A :0B0;V7C ?5@>:A8407>N, @503CT 7 4-0<V=>0=B8?V@8=>< (@50:FVO "@8=45@0). !:;04 @5035=BV2: R1 MES 1CD5@ (pH 6,5) 6,5 <<>;L/; N,N-1VA(4-AC;LD>1CB8;)-3-<5B8;0=V;V= 3 <<>;L/; >;V2V=V;AC;LD>=>20 :8A;>B0 50 <3 B5@ >;V5B8;5=-3;V:>;L-<5B8; 30 <;/; M03=VN E;>@84 2 <<>;L/; R2 MES 1CD5@ (pH 6,5) 50 <<>;L/; %>;5AB5@8=5AB5@070 (%) 5 :4/; %>;5AB5@8=>:A84070 (%) 20 :4/; 5@>:A84070 () 5 :4/; 4-0<V=>0=B8?V@8= (4-) 0,9 3/; 5B5@35=B 0,5 % >5DVFVT=B ?5@5@0EC=:C <<>;L/; = 0,026 E <3/4; >1>GV E0@0:B5@8AB8:8 =5 3V@H5 70: 'CB;82VABL: 1,9 <3/4; (0,049 <<>;L/;) V=V9=VABL: 4> 193 <3/4; (5,02 <<>;L/;) V0?07>= 28<V@N20==O: 1,9  193 <3/4; (0,049  5,02 <<>;L/;) #<>28 715@V30==O 2V4 +2 4> +8 C.?0:433696500-0-01>@0B>@=V @50:B82853395V?>?@>B5W= ) 8001V@ @5035=BV2 ?@87=0G5=89 4;O in vitro 287=0G5==O )-E>;5AB5@8=C (LDL) C A8@>20BFV V ?;07<V :@>2V ;N48=8. $0AC20==O: =5 <5=H5 R1: 2 x 30 <;, R2 : 2 E 10 <; @8=F8? <5B>4C 5B>4 4>72>;OT 287=0G8B8 )-E>;5AB5@8= 157 >A0465==O. 0 ?5@H><C 5B0?V ;V?>?@>B5W48 (), ) V EV;><V:@>=8) ?>2=VABN 3V4@>;V7CNBLAO V >:8A;NNBLAO 157 CB2>@5==O ?@>4C:BC, 2 B>9 G0A, O: ) T A5;5:B82=> 70E8I5=8<8. 0 4@C3><C 5B0?V ) 282V;L=NNBLAO 7 ?>40;LH8< 3V4@>;V7>< V >:8A;5==O< D5@<5=B0<8 E>;5AB5@8=5AB5@070 (%) V E>;5AB5@8=>:A84070 (%). #B2>@5=89 ?V4 G0A FL>3> ?@>F5AC ?5@5:8A 2>4=N 287=0G0TBLAO :V;L:VA=> 73V4=> <5B>4C "@8=45@0. !:;04 @5035=BV2: R1 MES-1CD5@ (pH 6,5) 50 <<>;L/; >;V2V=V;AC;LD>=V;>20 :8A;>B0 50 <3/; >;V5B8;5=3;V:>;L<5B8;>289 5B5@ 30 <;/; 4-0<V=>0=B8?V@8= 0,9 3/; %>;5AB5@8=5AB5@070 5 :4/; %>;5AB5@8=>:A84070 20 :4/; 5@>:A84070 () 5 :4/; 5B5@35=B R2 MES-1CD5@ (p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x 1 <;. !:;04 @5035=BV2: )/) 0;V1@0B>@ 2E1 <; >5DVFVT=B ?5@5@0EC=:C <3/4; x 0,026 = <<>;L/; V>;>3VG=89 <0B5@V0;, 7 O:8E 283>B>2;5=89 :0;V1@0B>@, 1C2 ?5@52V@5=89 =0 2V4ACB=VABL 0=B8BV; 4> 2V@CAC V<C=>45DVF8BC ;N48=8 (), 4> 2V@CAC 35?0B8BC ! 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